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Megestrol acetate

InhA, Func 595-33-5

Megestrol acetate (Megestrol acetate)

1 image

Catalog No. ABIN3221227

Quick Overview for Megestrol acetate (ABIN3221227)

Application

Inhibition Assay (InhA), Functional Studies (Func)

Purpose

Megestrol acetate is a progestogen with actions and uses similar to those of the progestogens in general. It also has anti-androgenic properties. It is given by mouth in the palliative treatment or as an adjunct to other therapy in endometrial carcinoma and in breast cancer. Megestrol acetate has been approved to treat anorexia and cachexia. (From Reynolds JEF(Ed): Martindale: The Extra Pharmacopoeia (electronic version). Micromedex, Inc, Englewood, CO, 1995)

Characteristics

Tradename: MEGACE
Source of Compound: semisynthetic, BDH-1298, SC-10363, 5071
Target: Glucocorticoid Receptor agonist, Estrogen/progestogen Receptor agonist
Receptor: Glucocorticoid receptor,Estrogen/progestogen Receptor

Purification

All the products are sent with COA, HPLC and NMR inspection report to guarantee the quality.

Purity

98 %

Formula

C24H32O4

Solubility

Water: 2 ?g/mL (at 37 °C)
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Application Notes

Optimal working dilution should be determined by the investigator.

Restrictions

For Research Use only
Format

Solid

Storage

-20 °C

Storage Comment

For the majority of compounds, they could be dissolved in DMSO or other organic solvent.
Their stock solution can be stored at -20°C for up to 3 months and aliquoted for sampling convenience.
Several freeze/thaw cycles should not damage the activity of our small molecule products.
However, in many instances the aqueous solutions of some compounds need to be made fresh and cannot be stored. For these compounds, their solution should be prepared just before use and stored no longer than 24 hours.

Expiry Date

24 months
Background

Endocrinology/ Hormones

Molecular Weight

384.51 g/mol

CAS-No

595-33-5

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